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-Structure paper
Title | Small Molecules Promote Selective Denaturation and Degradation of Tubulin Heterodimers through a Low-Barrier Hydrogen Bond. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 9159-9173, Year 2022 |
Publish date | Jun 19, 2020 (structure data deposition date) |
![]() | Yang, J. / Li, Y. / Qiu, Q. / Wang, R. / Yan, W. / Yu, Y. / Niu, L. / Pei, H. / Wei, H. / Ouyang, L. ...Yang, J. / Li, Y. / Qiu, Q. / Wang, R. / Yan, W. / Yu, Y. / Niu, L. / Pei, H. / Wei, H. / Ouyang, L. / Ye, H. / Xu, D. / Wei, Y. / Chen, Q. / Chen, L. |
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Methods | X-ray diffraction |
Resolution | 2.659 - 2.725 Å |
Structure data | ![]() PDB-7cda: ![]() PDB-7ce6: ![]() PDB-7ce8: ![]() PDB-7cek: |
Chemicals | ![]() ChemComp-GTP: ![]() ChemComp-MG: ![]() ChemComp-CA: ![]() ChemComp-GOL: ![]() ChemComp-GDP: ![]() ChemComp-MES: ![]() ChemComp-AEU: ![]() ChemComp-ACP: ![]() ChemComp-HOH: ![]() ChemComp-AF6: ![]() ChemComp-AEX: ![]() ChemComp-FW9: ![]() ChemComp-CL: |
Source |
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![]() | STRUCTURAL PROTEIN / tubulin inhibitor / tublin / STRUCTURAL PROTEIN-INHIBITOR COMPLEX |