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-Structure paper
Title | Design and Synthesis of TRAP1 Selective Inhibitors: H-Bonding with Asn171 Residue in TRAP1 Increases Paralog Selectivity. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 12, Page 1173-1180, Year 2021 |
Publish date | May 24, 2020 (structure data deposition date) |
![]() | Yang, S. / Yoon, N.G. / Kim, D. / Park, E. / Kim, S.Y. / Lee, J.H. / Lee, C. / Kang, B.H. / Kang, S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.5 - 3 Å |
Structure data | ![]() PDB-7c7b: ![]() PDB-7c7c: |
Chemicals | ![]() ChemComp-FJX: ![]() ChemComp-HOH: ![]() ChemComp-FK0: |
Source |
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![]() | CHAPERONE / TRAP1 / selectivity / mitochondria / Hsp90 / anticancer / drug / TRPA1 |