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-Structure paper
Title | Fragment-Based Discovery of Novel Allosteric MEK1 Binders. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 12, Page 302-308, Year 2021 |
Publish date | Dec 1, 2020 (structure data deposition date) |
Authors | Di Fruscia, P. / Edfeldt, F. / Shamovsky, I. / Collie, G.W. / Aagaard, A. / Barlind, L. / Borjesson, U. / Hansson, E.L. / Lewis, R.J. / Nilsson, M.K. ...Di Fruscia, P. / Edfeldt, F. / Shamovsky, I. / Collie, G.W. / Aagaard, A. / Barlind, L. / Borjesson, U. / Hansson, E.L. / Lewis, R.J. / Nilsson, M.K. / Oster, L. / Pemberton, J. / Ripa, L. / Storer, R.I. / Kack, H. |
External links | Acs Med. Chem. Lett. / PubMed:33603979 |
Methods | X-ray diffraction |
Resolution | 1.7 - 2.3 Å |
Structure data | PDB-7b3m: PDB-7b7r: PDB-7b94: PDB-7b9l: |
Chemicals | ChemComp-MG: ChemComp-ANP: ChemComp-SU5: ChemComp-SO4: ChemComp-HOH: ChemComp-T1K: ChemComp-PO4: ChemComp-T3W: ChemComp-T4N: ChemComp-GOL: |
Source |
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Keywords | TRANSFERASE / Kinase / allosteric / fragments |