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-Structure paper
Title | Bicyclic beta-Sheet Mimetics that Target the Transcriptional Coactivator beta-Catenin and Inhibit Wnt Signaling. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 60, Page 13937-13944, Year 2021 |
Publish date | Oct 23, 2020 (structure data deposition date) |
![]() | Wendt, M. / Bellavita, R. / Gerber, A. / Efrem, N.L. / van Ramshorst, T. / Pearce, N.M. / Davey, P.R.J. / Everard, I. / Vazquez-Chantada, M. / Chiarparin, E. ...Wendt, M. / Bellavita, R. / Gerber, A. / Efrem, N.L. / van Ramshorst, T. / Pearce, N.M. / Davey, P.R.J. / Everard, I. / Vazquez-Chantada, M. / Chiarparin, E. / Grieco, P. / Hennig, S. / Grossmann, T.N. |
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Methods | X-ray diffraction |
Resolution | 2.6 Å |
Structure data | ![]() PDB-7ar4: |
Chemicals | ![]() ChemComp-EPE: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
Source |
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![]() | SIGNALING PROTEIN / Wnt signaling / Peptide Inhibitor / Protein-Peptide Interaction |