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-Structure paper
Title | Design and Development of a Macrocyclic Series Targeting Phosphoinositide 3-Kinase delta. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 11, Page 1386-1391, Year 2020 |
Publish date | Jun 5, 2020 (structure data deposition date) |
Authors | Spencer, J.A. / Baldwin, I.R. / Barton, N. / Chung, C.W. / Convery, M.A. / Edwards, C.D. / Jamieson, C. / Mallett, D.N. / Rowedder, J.E. / Rowland, P. ...Spencer, J.A. / Baldwin, I.R. / Barton, N. / Chung, C.W. / Convery, M.A. / Edwards, C.D. / Jamieson, C. / Mallett, D.N. / Rowedder, J.E. / Rowland, P. / Thomas, D.A. / Hardy, C.J. |
External links | Acs Med. Chem. Lett. / PubMed:32676144 |
Methods | X-ray diffraction |
Resolution | 2.15 - 2.52 Å |
Structure data | PDB-6zaa: PDB-6zac: PDB-6zad: |
Chemicals | ChemComp-QD2: ChemComp-HOH: ChemComp-QDE: ChemComp-QDW: |
Source |
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Keywords | TRANSFERASE / Macrocycle / PI3K Delta / Thermodynamics |