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-Structure paper
Title | GSK973 Is an Inhibitor of the Second Bromodomains (BD2s) of the Bromodomain and Extra-Terminal (BET) Family. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 11, Page 1581-1587, Year 2020 |
Publish date | Jun 2, 2020 (structure data deposition date) |
![]() | Preston, A. / Atkinson, S.J. / Bamborough, P. / Chung, C.W. / Gordon, L.J. / Grandi, P. / Gray, J.R.J. / Harrison, L.A. / Lewis, A.J. / Lugo, D. ...Preston, A. / Atkinson, S.J. / Bamborough, P. / Chung, C.W. / Gordon, L.J. / Grandi, P. / Gray, J.R.J. / Harrison, L.A. / Lewis, A.J. / Lugo, D. / Messenger, C. / Michon, A.M. / Mitchell, D.J. / Prinjha, R.K. / Rioja, I. / Seal, J. / Taylor, S. / Thesmar, P. / Wall, I.D. / Watson, R.J. / Woolven, J.M. / Demont, E.H. |
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Methods | X-ray diffraction |
Resolution | 1.55 Å |
Structure data | ![]() PDB-6z8p: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-1PG: ![]() ChemComp-QC8: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / INHIBITOR / HISTONE / EPIGENETIC READER / BROMODOMAIN / BRD2 / BROMODOMAIN CONTAINING PROTEIN 2 / ANTAGONIST |