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-Structure paper
Title | Antitumor activity of a systemic STING-activating non-nucleotide cGAMP mimetic. |
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Journal, issue, pages | Science, Vol. 369, Page 993-999, Year 2020 |
Publish date | Jul 3, 2020 (structure data deposition date) |
![]() | Chin, E.N. / Yu, C. / Vartabedian, V.F. / Jia, Y. / Kumar, M. / Gamo, A.M. / Vernier, W. / Ali, S.H. / Kissai, M. / Lazar, D.C. ...Chin, E.N. / Yu, C. / Vartabedian, V.F. / Jia, Y. / Kumar, M. / Gamo, A.M. / Vernier, W. / Ali, S.H. / Kissai, M. / Lazar, D.C. / Nguyen, N. / Pereira, L.E. / Benish, B. / Woods, A.K. / Joseph, S.B. / Chu, A. / Johnson, K.A. / Sander, P.N. / Martinez-Pena, F. / Hampton, E.N. / Young, T.S. / Wolan, D.W. / Chatterjee, A.K. / Schultz, P.G. / Petrassi, H.M. / Teijaro, J.R. / Lairson, L.L. |
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Methods | X-ray diffraction |
Resolution | 1.77 - 2.49 Å |
Structure data | ![]() PDB-6xnn: ![]() PDB-6xnp: |
Chemicals | ![]() ChemComp-V67: ![]() ChemComp-HOH: ![]() ChemComp-GOL: ![]() ChemComp-EDO: |
Source |
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![]() | IMMUNE SYSTEM / Agonist / Complex / Closed Conformation / Immunity |