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| Title | An effective human uracil-DNA glycosylase inhibitor targets the open pre-catalytic active site conformation. |
|---|---|
| Journal, issue, pages | Prog. Biophys. Mol. Biol., Vol. 163, Page 143-159, Year 2021 |
| Publish date | Dec 18, 2019 (structure data deposition date) |
Authors | Nguyen, M.T. / Moiani, D. / Ahmed, Z. / Arvai, A.S. / Namjoshi, S. / Shin, D.S. / Fedorov, Y. / Selvik, E.J. / Jones, D.E. / Pink, J. ...Nguyen, M.T. / Moiani, D. / Ahmed, Z. / Arvai, A.S. / Namjoshi, S. / Shin, D.S. / Fedorov, Y. / Selvik, E.J. / Jones, D.E. / Pink, J. / Yan, Y. / Laverty, D.J. / Nagel, Z.D. / Tainer, J.A. / Gerson, S.L. |
External links | Prog. Biophys. Mol. Biol. / PubMed:33675849 |
| Methods | X-ray diffraction |
| Resolution | 1.8 Å |
| Structure data | ![]() PDB-6vba: |
| Chemicals | ![]() ChemComp-QU4: ![]() ChemComp-HOH: |
| Source |
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Keywords | HYDROLASE / GLYCOSYLASE / DNA REPAIR / URACIL REMOVAL FROM DNA / ALPHA/ BETA PROTEIN / GLYCOSIDASE |
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homo sapiens (human)
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