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-Structure paper
Title | Evaluating the Advantages of Using 3D-Enriched Fragments for Targeting BET Bromodomains. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 10, Page 1648-1654, Year 2019 |
Publish date | Nov 2, 2019 (structure data deposition date) |
![]() | Johnson, J.A. / Nicolaou, C.A. / Kirberger, S.E. / Pandey, A.K. / Hu, H. / Pomerantz, W.C.K. |
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Methods | X-ray diffraction |
Resolution | 1.307 - 1.51 Å |
Structure data | ![]() PDB-6uvj: ![]() PDB-6uvm: ![]() PDB-6uwx: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-DMS: ![]() ChemComp-QJ1: ![]() ChemComp-HOH: ![]() ChemComp-QJA: ![]() ChemComp-QKD: |
Source |
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![]() | GENE REGULATION/INHIBITOR / BRD4(D1) / inhibitor / GENE REGULATION-INHIBITOR complex |