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-Structure paper
Title | MET Tyrosine Kinase Inhibition Enhances the Antitumor Efficacy of an HGF Antibody. |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 16, Page 1269-1278, Year 2017 |
Publish date | Dec 19, 2016 (structure data deposition date) |
![]() | Farrell, P.J. / Matuszkiewicz, J. / Balakrishna, D. / Pandya, S. / Hixon, M.S. / Kamran, R. / Chu, S. / Lawson, J.D. / Okada, K. / Hori, A. ...Farrell, P.J. / Matuszkiewicz, J. / Balakrishna, D. / Pandya, S. / Hixon, M.S. / Kamran, R. / Chu, S. / Lawson, J.D. / Okada, K. / Hori, A. / Mizutani, A. / Iwata, H. / de Jong, R. / Hibner, B. / Vincent, P. |
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Methods | X-ray diffraction |
Resolution | 1.9 - 2.25 Å |
Structure data | ![]() PDB-5uab: ![]() PDB-5uad: ![]() PDB-6ubw: |
Chemicals | ![]() ChemComp-84M: ![]() ChemComp-GOL: ![]() ChemComp-CL: ![]() ChemComp-HOH: ![]() ChemComp-84P: ![]() ChemComp-84S: |
Source |
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![]() | TRANSFERASE/INHIBITOR / MET / Tyrosine Kinase / Inhibitor / Antitumor / TRANSFERASE-INHIBITOR complex / TRANSFERASE-TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |