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-Structure paper
Title | Pyrido[2,3-b][1,5]benzoxazepin-5(6H)-one derivatives as CDK8 inhibitors. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 201, Page 112443-112443, Year 2020 |
Publish date | Dec 12, 2019 (structure data deposition date) |
Authors | Martinez-Gonzalez, S. / Garcia, A.B. / Albarran, M.I. / Cebria, A. / Amezquita-Alves, A. / Garcia-Campos, F.J. / Martinez-Gago, J. / Martinez-Torrecuadrada, J. / Munoz, I. / Blanco-Aparicio, C. / Pastor, J. |
External links | Eur. J. Med. Chem. / PubMed:32599324 |
Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | PDB-6tpa: |
Chemicals | ChemComp-NZ8: ChemComp-FMT: ChemComp-NZ5: ChemComp-HOH: |
Source |
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Keywords | CELL CYCLE / Cell division Kinase Inhibitor |