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-Structure paper
Title | Discovery of Reversible Inhibitors of KDM1A Efficacious in Acute Myeloid Leukemia Models. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 11, Page 754-759, Year 2020 |
Publish date | Nov 11, 2019 (structure data deposition date) |
Authors | Romussi, A. / Cappa, A. / Vianello, P. / Brambillasca, S. / Cera, M.R. / Dal Zuffo, R. / Faga, G. / Fattori, R. / Moretti, L. / Trifiro, P. ...Romussi, A. / Cappa, A. / Vianello, P. / Brambillasca, S. / Cera, M.R. / Dal Zuffo, R. / Faga, G. / Fattori, R. / Moretti, L. / Trifiro, P. / Villa, M. / Vultaggio, S. / Cecatiello, V. / Pasqualato, S. / Dondio, G. / So, C.W.E. / Minucci, S. / Sartori, L. / Varasi, M. / Mercurio, C. |
External links | Acs Med. Chem. Lett. / PubMed:32435381 |
Methods | X-ray diffraction |
Resolution | 3.11 Å |
Structure data | PDB-6te1: |
Chemicals | ChemComp-N4K: ChemComp-FAD: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | OXIDOREDUCTASE / HISTONE DEMETHYLASE / INHIBITOR / COMPLEX |