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-Structure paper
Title | Cyclic boronates as versatile scaffolds for KPC-2 beta-lactamase inhibition. |
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Journal, issue, pages | Rsc Med Chem, Vol. 11, Page 491-496, Year 2020 |
Publish date | Nov 7, 2019 (structure data deposition date) |
Authors | Tooke, C.L. / Hinchliffe, P. / Krajnc, A. / Mulholland, A.J. / Brem, J. / Schofield, C.J. / Spencer, J. |
External links | Rsc Med Chem / PubMed:33479650 |
Methods | X-ray diffraction |
Resolution | 0.99 - 1.2 Å |
Structure data | PDB-6td0: PDB-6td1: |
Chemicals | ChemComp-4D6: ChemComp-GOL: ChemComp-SO4: ChemComp-HOH: ChemComp-KJK: |
Source |
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Keywords | ANTIMICROBIAL PROTEIN / inhibitor / boronate / beta-lactamase |