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-Structure paper
Title | Discovery of Highly Selective Inhibitors of Calmodulin-Dependent Kinases That Restore Insulin Sensitivity in the Diet-Induced Obesityin VivoMouse Model. |
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Journal, issue, pages | J. Med. Chem., Vol. 63, Page 6784-6801, Year 2020 |
Publish date | Oct 8, 2019 (structure data deposition date) |
Authors | Fromont, C. / Atzori, A. / Kaur, D. / Hashmi, L. / Greco, G. / Cabanillas, A. / Nguyen, H.V. / Jones, D.H. / Garzon, M. / Varela, A. ...Fromont, C. / Atzori, A. / Kaur, D. / Hashmi, L. / Greco, G. / Cabanillas, A. / Nguyen, H.V. / Jones, D.H. / Garzon, M. / Varela, A. / Stevenson, B. / Iacobini, G.P. / Lenoir, M. / Rajesh, S. / Box, C. / Kumar, J. / Grant, P. / Novitskaya, V. / Morgan, J. / Sorrell, F.J. / Redondo, C. / Kramer, A. / Harris, C.J. / Leighton, B. / Vickers, S.P. / Cheetham, S.C. / Kenyon, C. / Grabowska, A.M. / Overduin, M. / Berditchevski, F. / Weston, C.J. / Knapp, S. / Fischer, P.M. / Butterworth, S. |
External links | J. Med. Chem. / PubMed:32433887 |
Methods | X-ray diffraction |
Resolution | 1.484 - 1.55 Å |
Structure data | PDB-6t28: PDB-6t29: |
Chemicals | ChemComp-SO4: ChemComp-EDO: ChemComp-M92: ChemComp-HOH: ChemComp-M8Z: |
Source |
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Keywords | TRANSFERASE / Inhibitor / Complex / Kinase / Structural Genomics / Structural Genomics Consortium / SGC |