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-Structure paper
Title | Rapid Identification of Novel Allosteric PRC2 Inhibitors. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 14, Page 2134-2140, Year 2019 |
Publish date | Aug 1, 2019 (structure data deposition date) |
Authors | Read, J.A. / Tart, J. / Rawlins, P.B. / Gregson, C. / Jones, K. / Gao, N. / Zhu, X. / Tomlinson, R. / Code, E. / Cheung, T. ...Read, J.A. / Tart, J. / Rawlins, P.B. / Gregson, C. / Jones, K. / Gao, N. / Zhu, X. / Tomlinson, R. / Code, E. / Cheung, T. / Chen, H. / Kawatkar, S.P. / Bloecher, A. / Bagal, S. / O'Donovan, D.H. / Robinson, J. |
External links | Acs Chem. Biol. / PubMed:31525019 |
Methods | X-ray diffraction |
Resolution | 1.52 - 2 Å |
Structure data | PDB-6sfb: PDB-6sfc: |
Chemicals | ChemComp-L9W: ChemComp-GOL: ChemComp-HOH: ChemComp-CA: ChemComp-L9T: |
Source |
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Keywords | PROTEIN BINDING / Methyltransferase EED PRC2 epigenetic H3K27 WD40 Inhibitor |