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-Structure paper
Title | Crystal Structure of the first bromodomain of BRD4 in complex with a benzodiazepine ligand |
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Journal, issue, pages | To Be Published |
Publish date | Jun 20, 2019 (structure data deposition date) |
![]() | Picaud, S. / Traquete, R. / Bernardes, G.J.L. / Tobias, K. / von Delft, F. / Arrowsmith, C.H. / Edwards, A.M. / Bountra, C. / Filippakopoulos, P. / Structural Genomics Consortium (SGC) |
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Methods | X-ray diffraction |
Resolution | 1.1 Å |
Structure data | ![]() PDB-6s25: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-KSZ: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / BET / Bromodomain / RT53 / inhibitor / Structural Genomics / Structural Genomics Consortium / SGC |