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Title | Re-emerging Aspartic Protease Targets: Examining Cryptococcus neoformans Major Aspartyl Peptidase 1 as a Target for Antifungal Drug Discovery. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 6706-6719, Year 2021 |
Publish date | Mar 25, 2019 (structure data deposition date) |
![]() | Krystufek, R. / Sacha, P. / Starkova, J. / Brynda, J. / Hradilek, M. / Tloust'ova, E. / Grzymska, J. / Rut, W. / Boucher, M.J. / Drag, M. ...Krystufek, R. / Sacha, P. / Starkova, J. / Brynda, J. / Hradilek, M. / Tloust'ova, E. / Grzymska, J. / Rut, W. / Boucher, M.J. / Drag, M. / Majer, P. / Hajek, M. / Rezacova, P. / Madhani, H.D. / Craik, C.S. / Konvalinka, J. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.75 - 1.8 Å |
Structure data | ![]() PDB-6r5h: ![]() PDB-6r6a: |
Chemicals | ![]() ChemComp-PGE: ![]() ChemComp-PEG: ![]() ChemComp-EDO: ![]() ChemComp-SO4: ![]() ChemComp-NA: ![]() ChemComp-ACY: ![]() ChemComp-PG4: ![]() ChemComp-1PE: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / aspartyl protease / secreted / Cryptococcus neoformans |