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-Structure paper
Title | Discovery of a Potent and Selective Fragment-like Inhibitor of Methyllysine Reader Protein Spindlin 1 (SPIN1). |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 8996-9007, Year 2019 |
Publish date | Feb 14, 2019 (structure data deposition date) |
Authors | Xiong, Y. / Greschik, H. / Johansson, C. / Seifert, L. / Bacher, J. / Park, K.S. / Babault, N. / Martini, M. / Fagan, V. / Li, F. ...Xiong, Y. / Greschik, H. / Johansson, C. / Seifert, L. / Bacher, J. / Park, K.S. / Babault, N. / Martini, M. / Fagan, V. / Li, F. / Chau, I. / Christott, T. / Dilworth, D. / Barsyte-Lovejoy, D. / Vedadi, M. / Arrowsmith, C.H. / Brennan, P. / Fedorov, O. / Jung, M. / Farnie, G. / Liu, J. / Oppermann, U. / Schule, R. / Jin, J. |
External links | J. Med. Chem. / PubMed:31260300 |
Methods | X-ray diffraction |
Resolution | 1.6 Å |
Structure data | PDB-6qpl: |
Chemicals | ChemComp-MPD: ChemComp-DMS: ChemComp-JC5: ChemComp-GLY: ChemComp-PO4: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | CELL CYCLE / Epigenetics / Tudor domain / Methyl-Lysine / methyl-Arginine |