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-Structure paper
Title | Kallikrein 5 inhibitors identified through structure based drug design in search for a treatment for Netherton Syndrome. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 29, Page 821-825, Year 2019 |
Publish date | Jan 16, 2019 (structure data deposition date) |
![]() | White, G.V. / Edgar, E.V. / Holmes, D.S. / Lewell, X.Q. / Liddle, J. / Polyakova, O. / Smith, K.J. / Thorpe, J.H. / Walker, A.L. / Wang, Y. ...White, G.V. / Edgar, E.V. / Holmes, D.S. / Lewell, X.Q. / Liddle, J. / Polyakova, O. / Smith, K.J. / Thorpe, J.H. / Walker, A.L. / Wang, Y. / Young, R.J. / Hovnanian, A. |
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Methods | X-ray diffraction |
Resolution | 1.82 - 2.27 Å |
Structure data | ![]() PDB-6qh9: ![]() PDB-6qha: ![]() PDB-6qhb: ![]() PDB-6qhc: |
Chemicals | ![]() ChemComp-UNX: ![]() ChemComp-J2N: ![]() ChemComp-J3B: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-J2Q: ![]() ChemComp-J2W: ![]() ChemComp-135: ![]() ChemComp-DMS: |
Source |
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![]() | HYDROLASE / Protease / Inhibitor / Complex |