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-Structure paper
Title | Development of the First Low Nanomolar Liver Receptor Homolog-1 Agonist through Structure-guided Design. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 11022-11034, Year 2019 |
Publish date | Apr 29, 2019 (structure data deposition date) |
![]() | Mays, S.G. / Flynn, A.R. / Cornelison, J.L. / Okafor, C.D. / Wang, H. / Wang, G. / Huang, X. / Donaldson, H.N. / Millings, E.J. / Polavarapu, R. ...Mays, S.G. / Flynn, A.R. / Cornelison, J.L. / Okafor, C.D. / Wang, H. / Wang, G. / Huang, X. / Donaldson, H.N. / Millings, E.J. / Polavarapu, R. / Moore, D.D. / Calvert, J.W. / Jui, N.T. / Ortlund, E.A. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.004 - 2.23 Å |
Structure data | ![]() PDB-6oqx: ![]() PDB-6oqy: ![]() PDB-6or1: |
Chemicals | ![]() ChemComp-N1V: ![]() ChemComp-HOH: ![]() ChemComp-N2J: ![]() ChemComp-N27: |
Source |
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![]() | TRANSCRIPTION / Nuclear Hormone Receptor / agonist / Nuclear receptor / coactivator |