+Search query
-Structure paper
Title | Identification of Imidazo[1,2-b]pyridazine Derivatives as Potent, Selective, and Orally Active Tyk2 JH2 Inhibitors. |
---|---|
Journal, issue, pages | Acs Med. Chem. Lett., Vol. 10, Page 383-388, Year 2019 |
Publish date | Jan 25, 2019 (structure data deposition date) |
Authors | Liu, C. / Lin, J. / Moslin, R. / Tokarski, J.S. / Muckelbauer, J. / Chang, C. / Tredup, J. / Xie, D. / Park, H. / Li, P. ...Liu, C. / Lin, J. / Moslin, R. / Tokarski, J.S. / Muckelbauer, J. / Chang, C. / Tredup, J. / Xie, D. / Park, H. / Li, P. / Wu, D.R. / Strnad, J. / Zupa-Fernandez, A. / Cheng, L. / Chaudhry, C. / Chen, J. / Chen, C. / Sun, H. / Elzinga, P. / D'arienzo, C. / Gillooly, K. / Taylor, T.L. / McIntyre, K.W. / Salter-Cid, L. / Lombardo, L.J. / Carter, P.H. / Aranibar, N. / Burke, J.R. / Weinstein, D.S. |
External links | Acs Med. Chem. Lett. / PubMed:30891145 |
Methods | X-ray diffraction |
Resolution | 2.15 Å |
Structure data | PDB-6nsl: |
Chemicals | ChemComp-KZJ: ChemComp-SO4: ChemComp-HOH: |
Source |
|
Keywords | TRANSFERASE / KINASE |