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-Structure paper
Title | Identification and Optimization of Novel Small c-Abl Kinase Activators Using Fragment and HTS Methodologies. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 2154-2171, Year 2019 |
Publish date | Jan 17, 2019 (structure data deposition date) |
Authors | Simpson, G.L. / Bertrand, S.M. / Borthwick, J.A. / Campobasso, N. / Chabanet, J. / Chen, S. / Coggins, J. / Cottom, J. / Christensen, S.B. / Dawson, H.C. ...Simpson, G.L. / Bertrand, S.M. / Borthwick, J.A. / Campobasso, N. / Chabanet, J. / Chen, S. / Coggins, J. / Cottom, J. / Christensen, S.B. / Dawson, H.C. / Evans, H.L. / Hobbs, A.N. / Hong, X. / Mangatt, B. / Munoz-Muriedas, J. / Oliff, A. / Qin, D. / Scott-Stevens, P. / Ward, P. / Washio, Y. / Yang, J. / Young, R.J. |
External links | J. Med. Chem. / PubMed:30689376 |
Methods | X-ray diffraction |
Resolution | 1.86 - 2.33 Å |
Structure data | PDB-6npe: PDB-6npu: PDB-6npv: |
Chemicals | ChemComp-SO4: ChemComp-STI: ChemComp-KWD: ChemComp-2PE: ChemComp-HOH: ChemComp-KWV: ChemComp-GOL: ChemComp-KWP: |
Source |
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Keywords | TRANSFERASE / activator / kinase / allosteric / SIGNALING PROTEIN |