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-Structure paper
Title | A Potent and Selective Small-Molecule Degrader of STAT3 Achieves Complete Tumor Regression In Vivo. |
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Journal, issue, pages | Cancer Cell, Vol. 36, Page 498-511.e17, Year 2019 |
Publish date | Jan 4, 2019 (structure data deposition date) |
Authors | Bai, L. / Zhou, H. / Xu, R. / Zhao, Y. / Chinnaswamy, K. / McEachern, D. / Chen, J. / Yang, C.Y. / Liu, Z. / Wang, M. ...Bai, L. / Zhou, H. / Xu, R. / Zhao, Y. / Chinnaswamy, K. / McEachern, D. / Chen, J. / Yang, C.Y. / Liu, Z. / Wang, M. / Liu, L. / Jiang, H. / Wen, B. / Kumar, P. / Meagher, J.L. / Sun, D. / Stuckey, J.A. / Wang, S. |
External links | Cancer Cell / PubMed:31715132 |
Methods | X-ray diffraction |
Resolution | 2.7 - 3.15 Å |
Structure data | PDB-6njs: PDB-6nuq: |
Chemicals | ChemComp-KQV: ChemComp-HOH: |
Source |
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Keywords | transcription/transcription inhibitor / Stat3 / Activator / TRANSCRIPTION / transcription-transcription inhibitor complex |