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-Structure paper
Title | Structural basis of resistance of mutant RET protein-tyrosine kinase to its inhibitors nintedanib and vandetanib. |
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Journal, issue, pages | J. Biol. Chem., Vol. 294, Page 10428-10437, Year 2019 |
Publish date | Dec 17, 2018 (structure data deposition date) |
![]() | Terzyan, S.S. / Shen, T. / Liu, X. / Huang, Q. / Teng, P. / Zhou, M. / Hilberg, F. / Cai, J. / Mooers, B.H.M. / Wu, J. |
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Methods | X-ray diffraction |
Resolution | 1.87 - 1.99 Å |
Structure data | ![]() PDB-6ne7: ![]() PDB-6nec: ![]() PDB-6nja: |
Chemicals | ![]() ChemComp-FMT: ![]() ChemComp-AMP: ![]() ChemComp-HOH: ![]() ChemComp-XIN: ![]() ChemComp-ADE: |
Source |
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![]() | TRANSFERASE / oncogene / RET / Tyrosine Kinase / ATP-binding / Thyroid cancer / Non-small cell lung cancer / Nintedanib / complex |