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Structure paper

TitleTAS-120 Cancer Target Binding: Defining Reactivity and Revealing the First Fibroblast Growth Factor Receptor 1 (FGFR1) Irreversible Structure.
Journal, issue, pagesChemMedChem, Vol. 14, Page 494-500, Year 2019
Publish dateNov 5, 2018 (structure data deposition date)
AuthorsKalyukina, M. / Yosaatmadja, Y. / Middleditch, M.J. / Patterson, A.V. / Smaill, J.B. / Squire, C.J.
External linksChemMedChem / PubMed:30600916
MethodsX-ray diffraction
Resolution2 - 2.2 Å
Structure data

PDB-6mzq:
TAS-120 in reversible binding mode with FGFR1
Method: X-RAY DIFFRACTION / Resolution: 2 Å

PDB-6mzw:
TAS-120 covalent complex with FGFR1
Method: X-RAY DIFFRACTION / Resolution: 2.2 Å

Chemicals

ChemComp-TZ0:
1-[(3S)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1H-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one

ChemComp-HOH:
WATER

ChemComp-SO4:
SULFATE ION

Source
  • homo sapiens (human)
KeywordsTRANSFERASE/TRANSFERASE Inhibitor / FGFR1 / TAS-120 / inhibitor / complex / TRANSFERASE / TRANSFERASE-TRANSFERASE Inhibitor complex / covalent

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