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-Structure paper
Title | Molecular Basis for the N-Terminal Bromodomain-and-Extra-Terminal-Family Selectivity of a Dual Kinase-Bromodomain Inhibitor. |
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Journal, issue, pages | J. Med. Chem., Vol. 61, Page 9316-9334, Year 2018 |
Publish date | Sep 17, 2018 (structure data deposition date) |
Authors | Divakaran, A. / Talluri, S.K. / Ayoub, A.M. / Mishra, N.K. / Cui, H. / Widen, J.C. / Berndt, N. / Zhu, J.Y. / Carlson, A.S. / Topczewski, J.J. ...Divakaran, A. / Talluri, S.K. / Ayoub, A.M. / Mishra, N.K. / Cui, H. / Widen, J.C. / Berndt, N. / Zhu, J.Y. / Carlson, A.S. / Topczewski, J.J. / Schonbrunn, E.K. / Harki, D.A. / Pomerantz, W.C.K. |
External links | J. Med. Chem. / PubMed:30253095 |
Methods | X-ray diffraction |
Resolution | 1.6 - 1.74 Å |
Structure data | PDB-6mh1: PDB-6mh7: |
Chemicals | ChemComp-JQP: ChemComp-EDO: ChemComp-HOH: ChemComp-JQY: ChemComp-DMS: |
Source |
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Keywords | TRANSCRIPTION/TRANSCRIPTION INHIBITOR / CAP / HUNK1 / MCAP / PROTEIN BINDING-INHIBITOR COMPLEX / INHIBITOR / TRANSCRIPTION-INHIBITOR COMPLEX / Inflammation / MAP-Kinase Inhibition / TRANSCRIPTION-TRANSCRIPTION INHIBITOR complex / PROTEIN BINDING/INHIBITOR / bromodomain / 19F-NMR |