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-Structure paper
Title | CH7233163 Overcomes Osimertinib-Resistant EGFR-Del19/T790M/C797S Mutation. |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 19, Page 2288-2297, Year 2020 |
Publish date | Jan 27, 2020 (structure data deposition date) |
Authors | Kashima, K. / Kawauchi, H. / Tanimura, H. / Tachibana, Y. / Chiba, T. / Torizawa, T. / Sakamoto, H. |
External links | Mol. Cancer Ther. / PubMed:32943545 |
Methods | X-ray diffraction |
Resolution | 2.05 - 2.315 Å |
Structure data | PDB-6lub: PDB-6lud: |
Chemicals | ChemComp-EUX: ChemComp-HOH: ChemComp-YY3: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / PROTEIN KINASE / INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX / TRANSFERASE |