+Search query
-Structure paper
Title | Covalent Inhibitors Allosterically Block the Activation of Rho Family Proteins and Suppress Cancer Cell Invasion. |
---|---|
Journal, issue, pages | Adv Sci, Vol. 7, Page 2000098-2000098, Year 2020 |
Publish date | Sep 9, 2019 (structure data deposition date) |
Authors | Sun, Z. / Zhang, H. / Zhang, Y. / Liao, L. / Zhou, W. / Zhang, F. / Lian, F. / Huang, J. / Xu, P. / Zhang, R. ...Sun, Z. / Zhang, H. / Zhang, Y. / Liao, L. / Zhou, W. / Zhang, F. / Lian, F. / Huang, J. / Xu, P. / Zhang, R. / Lu, W. / Zhu, M. / Tao, H. / Yang, F. / Ding, H. / Chen, S. / Yue, L. / Zhou, B. / Zhang, N. / Tan, M. / Jiang, H. / Chen, K. / Liu, B. / Liu, C. / Dang, Y. / Luo, C. |
External links | Adv Sci / PubMed:32714746 |
Methods | X-ray diffraction |
Resolution | 1.454 - 1.981 Å |
Structure data | PDB-6kx2: PDB-6kx3: |
Chemicals | ChemComp-GDP: ChemComp-HOH: ChemComp-8ZO: |
Source |
|
Keywords | CELL INVASION / RHOA / GDP / Complex / inhibitor / covalent |