+Search query
-Structure paper
Title | Discovery, structural insight, and bioactivities of BY27 as a selective inhibitor of the second bromodomains of BET proteins. |
---|---|
Journal, issue, pages | Eur. J. Med. Chem., Vol. 182, Page 111633-111633, Year 2019 |
Publish date | May 5, 2019 (structure data deposition date) |
![]() | Chen, D. / Lu, T. / Yan, Z. / Lu, W. / Zhou, F. / Lyu, X. / Xu, B. / Jiang, H. / Chen, K. / Luo, C. / Zhao, Y. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.251 - 1.935 Å |
Structure data | ![]() PDB-6k04: ![]() PDB-6k05: |
Chemicals | ![]() ChemComp-CQF: ![]() ChemComp-HOH: ![]() ChemComp-MES: |
Source |
|
![]() | ANTITUMOR PROTEIN / Antitumor; BET proteins; Bromodomain inhibitor; Epigenetic readers |