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-Structure paper
Title | Stepwise Evolution of Fragment Hits against MAPK Interacting Kinases 1 and 2. |
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Journal, issue, pages | J. Med. Chem., Vol. 63, Page 621-637, Year 2020 |
Publish date | Mar 6, 2019 (structure data deposition date) |
![]() | Kwiatkowski, J. / Liu, B. / Pang, S. / Ahmad, N.H.B. / Wang, G. / Poulsen, A. / Yang, H. / Poh, Y.R. / Tee, D.H.Y. / Ong, E. ...Kwiatkowski, J. / Liu, B. / Pang, S. / Ahmad, N.H.B. / Wang, G. / Poulsen, A. / Yang, H. / Poh, Y.R. / Tee, D.H.Y. / Ong, E. / Retna, P. / Dinie, N. / Kwek, P. / Wee, J.L.K. / Manoharan, V. / Low, C.B. / Seah, P.G. / Pendharkar, V. / Sangthongpitag, K. / Joy, J. / Baburajendran, N. / Jansson, A.E. / Nacro, K. / Hill, J. / Keller, T.H. / Hung, A.W. |
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Methods | X-ray diffraction |
Resolution | 2.901 Å |
Structure data | ![]() PDB-6jlr: |
Chemicals | ![]() ChemComp-BV9: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Kinase / phosphorylation / inhibitor / MNK / kinase domain / TRANSFERASE / cancer / TRANSFERASE-TRANSFERASE INHIBITOR complex |