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-Structure paper
Title | Structure-Based Design and Synthesis of an Isozyme-Selective MTHFD2 Inhibitor with a Tricyclic Coumarin Scaffold. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 10, Page 893-898, Year 2019 |
Publish date | Feb 20, 2019 (structure data deposition date) |
![]() | Kawai, J. / Ota, M. / Ohki, H. / Toki, T. / Suzuki, M. / Shimada, T. / Matsui, S. / Inoue, H. / Sugihara, C. / Matsuhashi, N. ...Kawai, J. / Ota, M. / Ohki, H. / Toki, T. / Suzuki, M. / Shimada, T. / Matsui, S. / Inoue, H. / Sugihara, C. / Matsuhashi, N. / Matsui, Y. / Takaishi, S. / Nakayama, K. |
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Methods | X-ray diffraction |
Resolution | 2.25 - 2.5 Å |
Structure data | ![]() PDB-6jib: ![]() PDB-6jid: |
Chemicals | ![]() ChemComp-BQF: ![]() ChemComp-PO4: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-BQC: |
Source |
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![]() | OXIDOREDUCTASE / INHIBITOR / FOLATE / COFACTOR / DEHYDROGENASE |