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-Structure paper
Title | A novel series of human dihydroorotate dehydrogenase inhibitors discovered by in vitro screening: inhibition activity and crystallographic binding mode. |
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Journal, issue, pages | Febs Open Bio, Vol. 9, Page 1348-1354, Year 2019 |
Publish date | Jan 4, 2019 (structure data deposition date) |
![]() | Zeng, T. / Zuo, Z. / Luo, Y. / Zhao, Y. / Yu, Y. / Chen, Q. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 1.851 Å |
Structure data | ![]() PDB-6j3b: ![]() PDB-6j3c: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-FMN: ![]() ChemComp-ORO: ![]() ChemComp-B5O: ![]() ChemComp-LDA: ![]() ChemComp-DMS: ![]() ChemComp-ACT: ![]() ChemComp-CL: ![]() ChemComp-NA: ![]() ChemComp-HOH: ![]() ChemComp-B5X: |
Source |
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![]() | OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR / DHODH / Inhibitor / Complex / OXIDOREDUCTASE / OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex |