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-Structure paper
Title | Validation of Phosphodiesterase-10 as a Novel Target for Pulmonary Arterial Hypertension via Highly Selective and Subnanomolar Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 3707-3721, Year 2019 |
Publish date | Oct 10, 2018 (structure data deposition date) |
![]() | Huang, Y.Y. / Yu, Y.F. / Zhang, C. / Chen, Y. / Zhou, Q. / Li, Z. / Zhou, S. / Guo, L. / Wu, D. / Wu, Y. / Luo, H.B. |
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Methods | X-ray diffraction |
Resolution | 2.6 - 2.7 Å |
Structure data | ![]() PDB-6ijh: ![]() PDB-6iji: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-MG: ![]() ChemComp-AEO: ![]() ChemComp-HOH: ![]() ChemComp-AEL: |
Source |
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![]() | HYDROLASE/INHIBITOR / HYDROLASE-INHIBITOR complex |