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-Structure paper
Title | Discovery of an MLLT1/3 YEATS Domain Chemical Probe. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 57, Page 16302-16307, Year 2018 |
Publish date | Oct 2, 2018 (structure data deposition date) |
Authors | Moustakim, M. / Christott, T. / Monteiro, O.P. / Bennett, J. / Giroud, C. / Ward, J. / Rogers, C.M. / Smith, P. / Panagakou, I. / Diaz-Saez, L. ...Moustakim, M. / Christott, T. / Monteiro, O.P. / Bennett, J. / Giroud, C. / Ward, J. / Rogers, C.M. / Smith, P. / Panagakou, I. / Diaz-Saez, L. / Felce, S.L. / Gamble, V. / Gileadi, C. / Halidi, N. / Heidenreich, D. / Chaikuad, A. / Knapp, S. / Huber, K.V.M. / Farnie, G. / Heer, J. / Manevski, N. / Poda, G. / Al-Awar, R. / Dixon, D.J. / Brennan, P.E. / Fedorov, O. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:30288907 |
Methods | X-ray diffraction |
Resolution | 1.8 - 2.1 Å |
Structure data | PDB-6ht0: PDB-6ht1: |
Chemicals | ChemComp-SO4: ChemComp-EDO: ChemComp-GQ8: ChemComp-HOH: ChemComp-GQ5: |
Source |
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Keywords | TRANSCRIPTION / YEATS domain / ENL / MLLT1 / chemical probe / inhibitor / Structural Genomics / Structural Genomics Consortium / SGC |