+Search query
-Structure paper
Title | Type II Kinase Inhibitors Targeting Cys-Gatekeeper Kinases Display Orthogonality with Wild Type and Ala/Gly-Gatekeeper Kinases. |
---|---|
Journal, issue, pages | ACS Chem. Biol., Vol. 13, Page 2956-2965, Year 2018 |
Publish date | Sep 4, 2018 (structure data deposition date) |
Authors | Ocasio, C.A. / Warkentin, A.A. / McIntyre, P.J. / Barkovich, K.J. / Vesely, C. / Spencer, J. / Shokat, K.M. / Bayliss, R. |
External links | ACS Chem. Biol. / PubMed:30239186 |
Methods | X-ray diffraction |
Resolution | 2.13 - 2.4 Å |
Structure data | PDB-6hjj: PDB-6hjk: |
Chemicals | ChemComp-G7T: ChemComp-CL: ChemComp-ACT: ChemComp-PGF: ChemComp-HOH: ChemComp-G7W: ChemComp-SO4: |
Source |
|
Keywords | TRANSFERASE / Protein kinase / mitosis |