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-Structure paper
Title | 3,5,7-Substituted Pyrazolo[4,3- d]pyrimidine Inhibitors of Cyclin-Dependent Kinases and Their Evaluation in Lymphoma Models. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 4606-4623, Year 2019 |
Publish date | Jun 20, 2018 (structure data deposition date) |
![]() | Jorda, R. / Havlicek, L. / Sturc, A. / Tuskova, D. / Daumova, L. / Alam, M. / Skerlova, J. / Nekardova, M. / Perina, M. / Pospisil, T. ...Jorda, R. / Havlicek, L. / Sturc, A. / Tuskova, D. / Daumova, L. / Alam, M. / Skerlova, J. / Nekardova, M. / Perina, M. / Pospisil, T. / Siroka, J. / Urbanek, L. / Pachl, P. / Rezacova, P. / Strnad, M. / Klener, P. / Krystof, V. |
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Methods | X-ray diffraction |
Resolution | 2.15 Å |
Structure data | ![]() PDB-6gva: |
Chemicals | ![]() ChemComp-FCQ: ![]() ChemComp-EDO: ![]() ChemComp-CL: ![]() ChemComp-BR: ![]() ChemComp-PG4: ![]() ChemComp-SGM: ![]() ChemComp-PGE: ![]() ChemComp-HOH: |
Source |
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![]() | CELL CYCLE / cyclin-dependent kinase / pyrazolo[4 / 3-d]pyrimidine |