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-Structure paper
Title | High-affinity ligands of the colchicine domain in tubulin based on a structure-guided design. |
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Journal, issue, pages | Sci Rep, Vol. 8, Page 4242-4242, Year 2018 |
Publish date | Jan 24, 2018 (structure data deposition date) |
Authors | Bueno, O. / Estevez Gallego, J. / Martins, S. / Prota, A.E. / Gago, F. / Gomez-SanJuan, A. / Camarasa, M.J. / Barasoain, I. / Steinmetz, M.O. / Diaz, J.F. ...Bueno, O. / Estevez Gallego, J. / Martins, S. / Prota, A.E. / Gago, F. / Gomez-SanJuan, A. / Camarasa, M.J. / Barasoain, I. / Steinmetz, M.O. / Diaz, J.F. / Perez-Perez, M.J. / Liekens, S. / Priego, E.M. |
External links | Sci Rep / PubMed:29523799 |
Methods | X-ray diffraction |
Resolution | 2.098 - 2.148 Å |
Structure data | PDB-6fkj: PDB-6fkl: |
Chemicals | ChemComp-GTP: ChemComp-MG: ChemComp-CA: ChemComp-GOL: ChemComp-DLW: ChemComp-GDP: ChemComp-MES: ChemComp-PG4: ChemComp-ACP: ChemComp-HOH: ChemComp-DLK: |
Source |
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Keywords | CELL CYCLE / TUBULIN FOLD / CYTOSKELETON / MICROTUBULE |