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-Structure paper
Title | Design and Synthesis of Tetrahydroquinoxalines as Domain Selective BET Inhibitors |
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Journal, issue, pages | To Be Published |
Publish date | Jan 6, 2018 (structure data deposition date) |
![]() | Chung, C. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.83 Å |
Structure data | ![]() PDB-6ffd: |
Chemicals | ![]() ChemComp-D7T: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / INHIBITOR / HISTONE / EPIGENETIC READER / BROMODOMAIN / BRD4 / BROMODOMAIN CONTAINING PROTEIN 4 / ANTAGONIST |