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-Structure paper
Title | Targeting Ligandable Pockets on Plant Homeodomain (PHD) Zinc Finger Domains by a Fragment-Based Approach. |
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Journal, issue, pages | ACS Chem. Biol., Vol. 13, Page 915-921, Year 2018 |
Publish date | Dec 16, 2017 (structure data deposition date) |
Authors | Amato, A. / Lucas, X. / Bortoluzzi, A. / Wright, D. / Ciulli, A. |
External links | ACS Chem. Biol. / PubMed:29529862 |
Methods | X-ray diffraction |
Resolution | 1.9 - 2.7 Å |
Structure data | PDB-6fap: PDB-6fhq: PDB-6fhu: PDB-6fi0: PDB-6fi1: PDB-6fkp: |
Chemicals | ChemComp-ZN: ChemComp-PO4: ChemComp-D3H: ChemComp-GOL: ChemComp-HOH: ChemComp-DE5: ChemComp-K: ChemComp-DEW: |
Source |
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Keywords | TRANSCRIPTION / PHD / zinc finger / BAZ2B / BAZ2A / bromodomain / fragment / competition / epigenetic / PHD zinc finger / histone / 3-mer / epigenetic H3 / Fr 19 / Fr19 / ligandability / H3 |