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-Structure paper
Title | Structural and computational basis for potent inhibition of glutamate carboxypeptidase II by carbamate-based inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 27, Page 255-264, Year 2019 |
Publish date | Oct 27, 2017 (structure data deposition date) |
![]() | Barinka, C. / Novakova, Z. / Hin, N. / Bim, D. / Ferraris, D.V. / Duvall, B. / Kabarriti, G. / Tsukamoto, R. / Budesinsky, M. / Motlova, L. ...Barinka, C. / Novakova, Z. / Hin, N. / Bim, D. / Ferraris, D.V. / Duvall, B. / Kabarriti, G. / Tsukamoto, R. / Budesinsky, M. / Motlova, L. / Rojas, C. / Slusher, B.S. / Rokob, T.A. / Rulisek, L. / Tsukamoto, T. |
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Methods | X-ray diffraction |
Resolution | 1.52 - 1.68 Å |
Structure data | ![]() PDB-6ety: ![]() PDB-6ez9: ![]() PDB-6f5l: ![]() PDB-6fe5: |
Chemicals | ![]() ChemComp-NAG: ![]() ChemComp-ZN: ![]() ChemComp-CA: ![]() ChemComp-CL: ![]() ChemComp-BXK: ![]() ChemComp-HOH: ![]() ChemComp-C68: ![]() ChemComp-PGE: ![]() ChemComp-EDO: ![]() ChemComp-CQB: ![]() ChemComp-D6E: |
Source |
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![]() | HYDROLASE / glutamate carboxypeptidase II (GCPII); NAALADase; prostate-specific membrane antigen; phosphoramidate / glutamate carboxypeptidase II (GCPII); NAALADase; prostate-specific membrane antigen; |