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-Structure paper
Title | Identification and Structure-Guided Development of Pyrimidinone Based USP7 Inhibitors. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 9, Page 238-243, Year 2018 |
Publish date | Dec 1, 2017 (structure data deposition date) |
Authors | O'Dowd, C.R. / Helm, M.D. / Rountree, J.S.S. / Flasz, J.T. / Arkoudis, E. / Miel, H. / Hewitt, P.R. / Jordan, L. / Barker, O. / Hughes, C. ...O'Dowd, C.R. / Helm, M.D. / Rountree, J.S.S. / Flasz, J.T. / Arkoudis, E. / Miel, H. / Hewitt, P.R. / Jordan, L. / Barker, O. / Hughes, C. / Rozycka, E. / Cassidy, E. / McClelland, K. / Odrzywol, E. / Page, N. / Feutren-Burton, S. / Dvorkin, S. / Gavory, G. / Harrison, T. |
External links | ACS Med Chem Lett / PubMed:29541367 |
Methods | X-ray diffraction |
Resolution | 2.16 Å |
Structure data | PDB-6f5h: |
Chemicals | ChemComp-SO4: ChemComp-GOL: ChemComp-CQ5: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / USP7 / reversible / inhibitor / selective |