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-Structure paper
Title | 4-(Phenoxy) and 4-(benzyloxy)benzamides as potent and selective inhibitors of mono-ADP-ribosyltransferase PARP10/ARTD10. |
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Journal, issue, pages | Eur J Med Chem, Vol. 156, Page 93-102, Year 2018 |
Publish date | Sep 25, 2017 (structure data deposition date) |
Authors | Murthy, S. / Desantis, J. / Verheugd, P. / Maksimainen, M.M. / Venkannagari, H. / Massari, S. / Ashok, Y. / Obaji, E. / Nkizinkinko, Y. / Luscher, B. ...Murthy, S. / Desantis, J. / Verheugd, P. / Maksimainen, M.M. / Venkannagari, H. / Massari, S. / Ashok, Y. / Obaji, E. / Nkizinkinko, Y. / Luscher, B. / Tabarrini, O. / Lehtio, L. |
External links | Eur J Med Chem / PubMed:30006177 |
Methods | X-ray diffraction |
Resolution | 1.6 Å |
Structure data | PDB-6ek3: |
Chemicals | ChemComp-OUL: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / Inhibitor / OUL35 / SIGNALING PROTEIN |