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-Structure paper
Title | Biochemical Characterization and Structure-Based Mutational Analysis Provide Insight into the Binding and Mechanism of Action of Novel Aspartate Aminotransferase Inhibitors. |
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Journal, issue, pages | Biochemistry, Vol. 57, Page 6604-6614, Year 2018 |
Publish date | Jun 6, 2018 (structure data deposition date) |
![]() | Holt, M.C. / Assar, Z. / Beheshti Zavareh, R. / Lin, L. / Anglin, J. / Mashadova, O. / Haldar, D. / Mullarky, E. / Kremer, D.M. / Cantley, L.C. ...Holt, M.C. / Assar, Z. / Beheshti Zavareh, R. / Lin, L. / Anglin, J. / Mashadova, O. / Haldar, D. / Mullarky, E. / Kremer, D.M. / Cantley, L.C. / Kimmelman, A.C. / Stein, A.J. / Lairson, L.L. / Lyssiotis, C.A. |
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Methods | X-ray diffraction |
Resolution | 1.7 - 3 Å |
Structure data | ![]() PDB-6dna: ![]() PDB-6dnb: ![]() PDB-6dnd: |
Chemicals | ![]() ChemComp-PG4: ![]() ChemComp-PLP: ![]() ChemComp-HOH: ![]() ChemComp-GOL: ![]() ChemComp-PO4: |
Source |
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![]() | TRANSFERASE / Aspartate aminotransferase / Glutamate oxaloacetate transaminase 1 / GOT1 / PLP |