+Search query
-Structure paper
| Title | Discovery of a Highly Potent and Broadly Effective Epidermal Growth Factor Receptor and HER2 Exon 20 Insertion Mutant Inhibitor. |
|---|---|
| Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 57, Page 11629-11633, Year 2018 |
| Publish date | Apr 26, 2018 (structure data deposition date) |
Authors | Jang, J. / Son, J. / Park, E. / Kosaka, T. / Saxon, J.A. / De Clercq, D.J.H. / Choi, H.G. / Tanizaki, J. / Eck, M.J. / Janne, P.A. / Gray, N.S. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:29978938 |
| Methods | X-ray diffraction |
| Resolution | 2.537 Å |
| Structure data | ![]() PDB-6d8e: |
| Chemicals | ![]() ChemComp-FZP: ![]() ChemComp-HOH: |
| Source |
|
Keywords | Transferase/Transferase Inhibitor / EGFR / Inhibitor / SIGNALING PROTEIN / Transferase-Transferase Inhibitor complex |
Movie
Controller
Structure viewers
About Yorodumi Papers



Authors
External links


homo sapiens (human)
Keywords