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Title | Highly Potent and Selective Plasmin Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold Attenuate Fibrinolysis in Plasma. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 552-560, Year 2019 |
Publish date | Apr 17, 2018 (structure data deposition date) |
![]() | Swedberg, J.E. / Wu, G. / Mahatmanto, T. / Durek, T. / Caradoc-Davies, T.T. / Whisstock, J.C. / Law, R.H.P. / Craik, D.J. |
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Methods | X-ray diffraction |
Resolution | 1.32 - 2 Å |
Structure data | ![]() PDB-6d3x: ![]() PDB-6d3y: ![]() PDB-6d3z: ![]() PDB-6d40: |
Chemicals | ![]() ChemComp-HOH: ![]() ChemComp-SO4: ![]() ChemComp-GOL: |
Source |
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![]() | HYDROLASE / Protease / SFTI / complex / proteases / fibrinolysis / BLOOD CLOTTING |