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-Structure paper
Title | Identification of Thiourea-Based Inhibitors of the B-Cell Lymphoma 6 BTB Domain via NMR-Based Fragment Screening and Computer-Aided Drug Design. |
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Journal, issue, pages | J. Med. Chem., Vol. 61, Page 7573-7588, Year 2018 |
Publish date | Jan 10, 2018 (structure data deposition date) |
Authors | Cheng, H. / Linhares, B.M. / Yu, W. / Cardenas, M.G. / Ai, Y. / Jiang, W. / Winkler, A. / Cohen, S. / Melnick, A. / MacKerell Jr., A. ...Cheng, H. / Linhares, B.M. / Yu, W. / Cardenas, M.G. / Ai, Y. / Jiang, W. / Winkler, A. / Cohen, S. / Melnick, A. / MacKerell Jr., A. / Cierpicki, T. / Xue, F. |
External links | J. Med. Chem. / PubMed:29969259 |
Methods | X-ray diffraction |
Resolution | 1.46092157578 - 2.53170577659 Å |
Structure data | PDB-6c3l: PDB-6c3n: PDB-6cq1: |
Chemicals | ChemComp-EGP: ChemComp-HOH: ChemComp-EHY: ChemComp-F8J: |
Source |
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Keywords | protein binding/inhibitor / Inhibitor / protein-protein interaction / PROTEIN BINDING / protein binding-inhibitor complex / TRANSCRIPTION/Inhibitor / TRANSCRIPTION-Inhibitor complex / Protein protein inhibitor |