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Title | Selective, Small-Molecule Co-Factor Binding Site Inhibition of a Su(var)3-9, Enhancer of Zeste, Trithorax Domain Containing Lysine Methyltransferase. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 7669-7683, Year 2019 |
Publish date | Feb 5, 2018 (structure data deposition date) |
Authors | Taylor, A.P. / Swewczyk, M. / Kennedy, S. / Trush, V.V. / Wu, H. / Zeng, H. / Dong, A. / Ferreira de Freitas, R. / Tatlock, J. / Kumpf, R.A. ...Taylor, A.P. / Swewczyk, M. / Kennedy, S. / Trush, V.V. / Wu, H. / Zeng, H. / Dong, A. / Ferreira de Freitas, R. / Tatlock, J. / Kumpf, R.A. / Wythes, M. / Casimiro-Garcia, A. / Denny, R.A. / Parikh, M.D. / Li, F. / Barsyte-Lovejoy, D. / Schapira, M. / Vedadi, M. / Brown, P.J. / Arrowsmith, C.H. / Owen, D.R. |
External links | J. Med. Chem. / PubMed:31415173 |
Methods | X-ray diffraction |
Resolution | 2.55 Å |
Structure data | PDB-6cby: |
Chemicals | ChemComp-ZN: ChemComp-EW4: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/INHIBITOR / SMYD2 MTF9975 inhibitor / Structural Genomics / Structural Genomics Consortium / SGC / TRANSFERASE-INHIBITOR complex |