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Title | Design, synthesis, in vitro activity and crystallisation of novel N-isopropyl-N-hydroxyoxamate derivatives as ketol-acid reductosiomerase (KARI) inhibitor |
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Journal, issue, pages | To Be Published |
Publish date | Jan 16, 2018 (structure data deposition date) |
![]() | Kandale, A. / Patel, K.M. / Zheng, S. / You, L. / Guddat, L.W. / Schenk, G. / Schembri, M.A. / McGeary, R.P. |
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Methods | X-ray diffraction |
Resolution | 1.673 Å |
Structure data | ![]() PDB-6c5n: |
Chemicals | ![]() ChemComp-NDP: ![]() ChemComp-MG: ![]() ChemComp-EN4: ![]() ChemComp-81B: ![]() ChemComp-IMD: ![]() ChemComp-HOH: |
Source |
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![]() | OXIDOREDUCTASE / ketol-acid reductoisomerase / isomerase / inhibitor |