+Search query
-Structure paper
Title | Structure Based Design of a Grp94-Selective Inhibitor: Exploiting a Key Residue in Grp94 To Optimize Paralog-Selective Binding. |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 61, Page 2793-2805, Year 2018 |
Publish date | May 26, 2017 (structure data deposition date) |
Authors | Que, N.L.S. / Crowley, V.M. / Duerfeldt, A.S. / Zhao, J. / Kent, C.N. / Blagg, B.S.J. / Gewirth, D.T. |
External links | J. Med. Chem. / PubMed:29528635 |
Methods | X-ray diffraction |
Resolution | 1.792 - 2.895 Å |
Structure data | PDB-5vyy: PDB-5wmt: PDB-6baw: PDB-6c91: PDB-6ceo: |
Chemicals | ChemComp-9QY: ChemComp-FMT: ChemComp-EDO: ChemComp-MG: ChemComp-NA: ChemComp-HOH: ChemComp-D57: ChemComp-PO4: ChemComp-SO4: ChemComp-EQD: |
Source |
|
Keywords | CHAPERONE/INHIBITOR / chaperone / chaperone-inhibitor / CHAPERONE-INHIBITOR complex / Inhibitor / Complex / endoplasmin |