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-Structure paper
Title | Novel K-Ras G12C Switch-II Covalent Binders Destabilize Ras and Accelerate Nucleotide Exchange. |
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Journal, issue, pages | J Chem Inf Model, Vol. 58, Page 464-471, Year 2018 |
Publish date | Aug 22, 2017 (structure data deposition date) |
Authors | Nnadi, C.I. / Jenkins, M.L. / Gentile, D.R. / Bateman, L.A. / Zaidman, D. / Balius, T.E. / Nomura, D.K. / Burke, J.E. / Shokat, K.M. / London, N. |
External links | J Chem Inf Model / PubMed:29320178 |
Methods | X-ray diffraction |
Resolution | 1.75 Å |
Structure data | PDB-6ark: |
Chemicals | ChemComp-GDP: ChemComp-MG: ChemComp-BQD: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | signaling protein/inhibitor / DOCKovalent / covalent docking / K-Ras G12C / covalent inhibitors / covalent fragments / SIGNALING PROTEIN / signaling protein-inhibitor complex |